SCHEMBL20249117

SCHEMBL20249117

CC(C)(C)c1ccc(N2CCC(C(=O)O)CC2)cn1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.49
NOTUM Q6P988 12/20 0.47
KDM4E B2RXH2 2/20 0.47
CYP2C19 P33261 1/20 0.47
CHRM4 P08173 1/20 0.44
USP2 O75604 1/20 0.43
HPGD P15428 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HSD17B10 Q99714 1/20 0.43
AKR1C3 P42330 1/20 0.43
NEK2 P51955 1/20 0.43
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31381230 0.86 HRH3 (0.60) HRH3NOTUMKDM4ECYP2C19CHRM4
SCHEMBL17714317 0.86 HRH3 (0.60) HRH3NOTUMKDM4ECYP2C19CHRM4
SCHEMBL237457 0.82 KDM4E (0.55) NOTUMKDM4ECYP2C19USP2HPGD
SCHEMBL20249098 0.82 MAPT (0.46) HRH3
SCHEMBL20249226 0.81 MAPT (0.45) HRH3CHRM4
SCHEMBL20255191 0.80 HRH4 (0.43) HRH3
SCHEMBL31647908 0.80 NOTUM (0.67) HRH3NOTUMCHRM4
SCHEMBL20249116 0.78 ABL1 (0.43) HRH3
SCHEMBL20037680 0.78 NOTUM (0.50) NOTUMKDM4ECYP2C19USP2HPGD
SCHEMBL16398202 0.78 NEK2 (0.52) NOTUMKDM4ECYP2C19USP2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF TEIJIN PHARMA LIMITED (JP) 2018-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF CDK4, CDK6, CDK16 HRH3 2304/4885NOTUM 2845/4885KDM4E 470/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.