SCHEMBL20258487

SCHEMBL20258487

CNCCCC[C@@H]1CCN(c2c(F)cc3c(=O)c(C(=O)O)cn(Cc4ccc5ccccc5c4)c3c2OC)C1

nearest known ligand 0.79

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 12/20 0.79
KCNH2 Q12809 3/20 0.52
KDM4E B2RXH2 4/20 0.46
ALDH1A1 P00352 3/20 0.46
POLB P06746 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
LMNA P02545 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HPGD P15428 3/20 0.44
PRKD3 O94806 1/20 0.44
ALOX15 P16050 1/20 0.44
OPRM1 P35372 1/20 0.44
CLK2 P49760 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20258365 0.93 TOP1 (0.84) TOP1KCNH2KDM4EALDH1A1POLB
SCHEMBL20258407 0.92 TOP1 (0.78) TOP1KCNH2KDM4EALDH1A1POLB
SCHEMBL21787290 0.90 TOP1 (0.90) TOP1KCNH2KDM4EALDH1A1POLB
SCHEMBL20258379 0.89 TOP1 (0.88) TOP1KCNH2KDM4EALDH1A1POLB
SCHEMBL20258411 0.89 TOP1 (0.88) TOP1KCNH2KDM4EALDH1A1POLB
SCHEMBL20258486 0.89 TOP1 (0.71) TOP1KCNH2KDM4EALDH1A1POLB
SCHEMBL20242745 0.88 TOP1 (1.00) TOP1KCNH2KDM4EALDH1A1POLB
SCHEMBL20258348 0.88 TOP1 (1.00) TOP1KCNH2KDM4EALDH1A1POLB
SCHEMBL20242743 0.88 TOP1 (1.00) TOP1KCNH2KDM4EALDH1A1POLB
SCHEMBL21786930 0.84 TOP1 (0.81) TOP1KCNH2KDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018107112-A1 QUINOLONE-BASED COMPOUNDS WITH ANTICANCER ACTIVITY UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2018-06-14 WO disclosed