SCHEMBL2025875

SCHEMBL2025875

CN(c1cc(-c2ncc([C@](C)(NC(=O)O)C(c3ccccc3)C(C)(C)C)o2)cc(Cl)n1)S(C)(=O)=O

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 6/20 0.39
BACE2 Q9Y5Z0 3/20 0.32
MAPK1 P28482 1/20 0.32
P2RY12 Q9H244 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2023991 0.87 BACE1 (0.41) BACE1BACE2MAPK1
SCHEMBL4945797 0.82 BACE1 (0.44) BACE1BACE2
SCHEMBL4947313 0.78 BACE1 (0.37) BACE1BACE2MAPK1
SCHEMBL2027660 0.76 BACE1 (0.36) BACE1BACE2MAPK1
SCHEMBL12578541 0.76 BACE1 (0.42) BACE1BACE2
SCHEMBL4939179 0.72 BACE1 (0.49) BACE1BACE2
SCHEMBL4942412 0.72 BACE1 (0.49) BACE1BACE2
SCHEMBL2026306 0.71 BACE1 (0.38) BACE1BACE2MAPK1
SCHEMBL13269914 0.70 BACE1 (0.40) BACE1BACE2
SCHEMBL2023118 0.69 BACE1 (0.37) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7968571-B2 2,4,6-substituted pyridyl derivative compounds useful as beta-secretase inhibitors for the treatment of Alzheimer's Disease Merck, Sharp & Dohme, Corp. (US) 2011-06-28 US disclosed