SCHEMBL20277652

SCHEMBL20277652

Cc1cc(C(=O)N2Cc3cn[nH]c3Nc3ccccc32)ccc1CN

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 13/20 0.52
OXTR P30559 11/20 0.52
AVPR2 P30518 8/20 0.52
CHRM2 P08172 1/20 0.43
CHRM4 P08173 1/20 0.43
CHRM5 P08912 1/20 0.43
CHRM3 P20309 1/20 0.43
DRD3 P35462 1/20 0.43
OPRK1 P41145 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HTT P42858 1/20 0.39
BRD4 O60885 1/20 0.39
BRD2 P25440 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2130122 0.82 AVPR1A (0.74) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL6201929 0.76 BRD4 (0.60) AVPR1AOXTRAVPR2ALDH1A1LMNA
SCHEMBL5570643 0.74 AVPR1A (0.65) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL2704576 0.74 AVPR1A (0.61) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL18917221 0.72 AVPR1A (0.63) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL2129142 0.72 AVPR1A (0.61) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL5567012 0.72 AVPR1A (0.63) AVPR1AOXTRAVPR2CHRM2CHRM4
Hydrochloric Acid SCHEMBL5270039 0.72 AVPR2 (0.56) AVPR1AOXTRAVPR2
SCHEMBL18944536 0.72 AVPR1A (0.80) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL9961437 0.72 AVPR1A (0.72) AVPR1AOXTRAVPR2CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018107216-A1 NON-PEPTIDE OXYTOCIN RECEPTOR AGONISTS THE UNIVERSITY OF SYDNEY (AU) 2018-06-21 WO disclosed