SCHEMBL20283113

SCHEMBL20283113

CC(C)(C)OC(=O)N1CC(C(=N)N)C(c2cccc(Cl)c2)C1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 9/20 0.53
TACR1 P25103 2/20 0.46
RORC P51449 1/20 0.44
MC4R P32245 2/20 0.44
STS P08842 2/20 0.43
SLC9A1 P19634 1/20 0.42
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
GRM5 P41594 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20283114 0.89 PDE4B (0.53) PDE4BTACR1RORCMC4RSTS
SCHEMBL16780016 0.88 PDE4B (0.57) PDE4BTACR1RORCMC4RSTS
SCHEMBL13858719 0.88 PDE4B (0.57) PDE4BTACR1RORCMC4RSTS
SCHEMBL16780015 0.88 PDE4B (0.57) PDE4BTACR1RORCMC4RSTS
SCHEMBL528139 0.84 DPP4 (0.51) PDE4BTACR1RORCMC4RSTS
SCHEMBL4008250 0.80 PDE4B (0.57) PDE4BTACR1RORCSTSTP53
SCHEMBL14498551 0.80 PDE4B (0.57) PDE4BTACR1RORCSTSTP53
SCHEMBL14495628 0.80 PDE4B (0.57) PDE4BTACR1RORCSTSTP53
SCHEMBL20757065 0.80 TP53 (0.52) PDE4BRORCSTSTP53MAPT
SCHEMBL31171241 0.79 PDE4B (0.59) PDE4BTACR1RORCMC4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3555065-B1 COMPOUNDS AS MODULATORS OF ROR GAMMA BOEHRINGER INGELHEIM INT (DE) 2021-02-24 EP disclosed
WO-2018111803-A1 COMPOUNDS AS MODULATORS OF ROR GAMMA BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-06-21 WO disclosed