SCHEMBL20311191

SCHEMBL20311191

CC(C)(C)S(=O)(=O)c1ccc(NC(=N)c2c(N)cc[nH]c2=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.42
JAK2 O60674 15/20 0.37
JAK1 P23458 15/20 0.37
ATR Q13535 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20245973 0.86 EGFR (0.44) EGFRJAK2JAK1
SCHEMBL20311056 0.84 JAK2 (0.40) EGFRJAK2JAK1CA1CA2
SCHEMBL20246302 0.80 EGFR (0.41) EGFR
SCHEMBL20311130 0.78 EGFR (0.44) EGFRJAK2JAK1CA12CA1
SCHEMBL20246267 0.78 EGFR (0.43) EGFR
SCHEMBL16623589 0.78 EGFR (0.43) EGFRJAK2ATR
SCHEMBL20246564 0.78 PTGS1 (0.43) EGFRCA12CA1CA2CA9
SCHEMBL20246361 0.77 EGFR (0.39) EGFR
SCHEMBL20311022 0.75 EGFR (0.42) EGFRJAK2JAK1CA12CA1
SCHEMBL20310858 0.75 EGFR (0.40) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2976339-B1 GEMINALLY SUBSTITUTED CYANOETHYLPYRAZOLO PYRIDONES AS JANUS KINASE INHIBITORS MERCK SHARP & DOHME (US) 2018-06-27 EP disclosed