Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | CACNA1F | O60840 | 5/20 | 0.36 |
| ▸ | CACNA1D | Q01668 | 5/20 | 0.36 |
| ▸ | CACNA1S | Q13698 | 5/20 | 0.36 |
| ▸ | CACNA1C | Q13936 | 5/20 | 0.36 |
| ▸ | HTT | P42858 | 2/20 | 0.35 |
| ▸ | XBP1 | P17861 | 1/20 | 0.34 |
| ▸ | ADRA1D | P25100 | 1/20 | 0.34 |
| ▸ | ADRA1A | P35348 | 1/20 | 0.34 |
| ▸ | ADRA1B | P35368 | 1/20 | 0.34 |
| ▸ | ACHE | P22303 | 2/20 | 0.33 |
| ▸ | MBTPS1 | Q14703 | 1/20 | 0.32 |
| ▸ | TP53 | P04637 | 1/20 | 0.32 |
| ▸ | MAPT | P10636 | 1/20 | 0.32 |
| ▸ | ALOX15 | P16050 | 1/20 | 0.32 |
| ▸ | TSHR | P16473 | 1/20 | 0.32 |
| ▸ | MAPK1 | P28482 | 1/20 | 0.32 |
| ▸ | NPSR1 | Q6W5P4 | 1/20 | 0.32 |
| ▸ | MEN1 | O00255 | 1/20 | 0.32 |
| ▸ | LMNA | P02545 | 1/20 | 0.32 |
| ▸ | GAA | P10253 | 1/20 | 0.32 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL20328325 | 0.88 | CACNA1F (0.40) | CACNA1FCACNA1DCACNA1SCACNA1CHTT | |
| SCHEMBL5568116 | 0.84 | CACNA1F (0.40) | CACNA1FCACNA1DCACNA1SCACNA1CHTT | |
| SCHEMBL5568028 | 0.79 | HTT (0.40) | CACNA1FCACNA1DCACNA1SCACNA1CHTT | |
| SCHEMBL5569023 | 0.79 | HTT (0.42) | CACNA1FCACNA1DCACNA1SCACNA1CHTT | |
| SCHEMBL5567175 | 0.79 | HTT (0.40) | CACNA1FCACNA1DCACNA1SCACNA1CHTT | |
| SCHEMBL5568485 | 0.78 | HTT (0.39) | CACNA1FCACNA1DCACNA1SCACNA1CHTT | |
| SCHEMBL5562836 | 0.78 | CACNA1F (0.55) | CACNA1FCACNA1DCACNA1SCACNA1CMAPT | |
| SCHEMBL5563157 | 0.77 | HTT (0.39) | CACNA1FCACNA1DCACNA1SCACNA1CHTT | |
| SCHEMBL5563112 | 0.77 | CACNA1F (0.40) | CACNA1FCACNA1DCACNA1SCACNA1CHTT | |
| SCHEMBL20328168 | 0.77 | CACNA1F (0.40) | CACNA1FCACNA1DCACNA1SCACNA1CHTT |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| WO-2018118101-A1 | T-TYPE CALCIUM CHANNEL MODULATORS AND METHODS OF USE THEREOF | PRAXIS PRECISION MEDICINES, INC. (US) | 2018-06-28 | — | — | WO | disclosed |