SCHEMBL20329862

SCHEMBL20329862

CNc1cc(N)ccc1-c1ccc(C(F)(F)F)nc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.48
PIK3CA P42336 2/20 0.48
PI4KB Q9UBF8 2/20 0.48
MAP4K4 O95819 2/20 0.48
MINK1 Q8N4C8 1/20 0.48
PIK3CD O00329 1/20 0.41
PIK3CB P42338 1/20 0.41
PI4KA P42356 1/20 0.41
PIK3CG P48736 1/20 0.41
PDE10A Q9Y233 1/20 0.41
MTOR P42345 2/20 0.40
FEN1 P39748 5/20 0.38
ALOX5AP P20292 3/20 0.38
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
GLA P06280 1/20 0.37
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37
TSHR P16473 1/20 0.37
TRPV4 Q9HBA0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7085072 0.78 KCNH2 (0.50) KCNH2PIK3CAPI4KBMAP4K4MINK1
SCHEMBL21497167 0.77 KCNH2 (0.49) KCNH2PIK3CAPI4KBMAP4K4MINK1
SCHEMBL25010664 0.76 KCNH2 (0.47) KCNH2PIK3CAPI4KBMAP4K4MINK1
SCHEMBL21071606 0.75 ALOX5AP (0.46) KCNH2PIK3CAPI4KBMAP4K4MINK1
SCHEMBL3786718 0.75 CYP3A4 (0.40) MAP4K4FEN1GLAPOLBGAA
SCHEMBL23951820 0.73 PIK3CA (0.53) KCNH2PIK3CAPI4KBMAP4K4MINK1
SCHEMBL21497106 0.72 KCNH2 (0.45) KCNH2PIK3CAPI4KBMAP4K4MINK1
SCHEMBL17407893 0.71 FEN1 (0.54) KCNH2PIK3CAPI4KBMAP4K4MINK1
SCHEMBL20329375 0.70 TSHR (0.41) FEN1ALOX5APGLAPOLBGAA
SCHEMBL21135415 0.70 KCNH2 (0.41) KCNH2PIK3CAPI4KBMAP4K4MINK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018114783-A1 TETRAZOLE CONTAINING COMPOUNDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-06-28 WO disclosed