SCHEMBL2033253

SCHEMBL2033253

Nc1ccnc(C2CCCNC2)n1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 2/20 0.46
CCNA2 P20248 2/20 0.46
CDK2 P24941 2/20 0.46
CCNA1 P78396 2/20 0.46
CCNT1 O60563 1/20 0.44
CDK9 P50750 1/20 0.44
ROCK1 Q13464 2/20 0.40
ROCK2 O75116 1/20 0.40
KCNH2 Q12809 1/20 0.40
ADORA2A P29274 1/20 0.39
MAPK8 P45983 1/20 0.39
BTK Q06187 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28245182 1.00 CHEK1 (0.46) CHEK1CCNA2CDK2CCNA1CCNT1
SCHEMBL28063327 0.90 HRH3 (0.42) CHEK1CCNA2CDK2CCNA1CCNT1
SCHEMBL30260114 0.81 FEN1 (0.39) KCNH2
SCHEMBL1221900 0.81 FEN1 (0.39) KCNH2
SCHEMBL1831010 0.81 BACE1 (0.41) KCNH2
SCHEMBL15587840 0.81 MAP3K12 (0.43) CHEK1CCNA2CDK2CCNA1MAPK8
SCHEMBL2034798 0.80 CHEK1 (0.47) CHEK1CCNA2CDK2CCNA1
SCHEMBL3567520 0.80 MKNK1 (0.44) CCNT1CDK9ROCK1
SCHEMBL23667387 0.80 BACE1 (0.44) KCNH2
Hydrochloric Acid SCHEMBL20292168 0.79 MKNK1 (0.43) CCNT1CDK9ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133657-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AND THEIR USE IN TREATMENT, AMELIORATION OR PREVENTION OF INFLUENZA SAVIRA PHARMACEUTICALS GMBH (AT) 2017-08-10 WO disclosed
EP-2516436-A1 IMIDAZOPYRIDINE DERIVATIVES AS JAK INHIBITORS Almirall S.A. (ES) 2012-10-31 EP disclosed
WO-2011076419-A1 IMIDAZOPYRIDINE DERIVATIVES AS JAK INHIBITORS ALMIRALL, S.A. (ES) 2011-06-30 WO disclosed