SCHEMBL20344703

SCHEMBL20344703

CCCN1C(=O)CCc2cc(NS(=O)(=O)Cc3ccc(Cl)cc3C)ccc21

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.42
BRD4 O60885 2/20 0.41
CREBBP Q92793 1/20 0.41
HDAC1 Q13547 3/20 0.39
HDAC8 Q9BY41 3/20 0.39
HDAC6 Q9UBN7 3/20 0.39
TRIM24 O15164 4/20 0.38
NPY5R Q15761 1/20 0.37
ATAD2 Q6PL18 1/20 0.37
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
P2RX7 Q99572 1/20 0.36
TP53 P04637 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
PKM P14618 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22692407 0.89 IDH1 (0.43) IDH1BRD4CREBBPHDAC1HDAC8
SCHEMBL20344731 0.84 BRD4 (0.41) BRD4CREBBPHDAC1HDAC8HDAC6
SCHEMBL30803804 0.82 BRD4 (0.41) BRD4CREBBPHDAC1HDAC8HDAC6
SCHEMBL20344748 0.82 BRD4 (0.41) BRD4CREBBPHDAC1HDAC8HDAC6
SCHEMBL20344770 0.82 BRD4 (0.41) BRD4CREBBPHDAC1HDAC8HDAC6
SCHEMBL15298954 0.81 BRD4 (0.44) BRD4CREBBPHDAC1HDAC8HDAC6
SCHEMBL20344751 0.78 BRD4 (0.41) BRD4CREBBPHDAC1HDAC8HDAC6
SCHEMBL29424983 0.78 BRD4 (0.42) IDH1BRD4CREBBPHDAC1HDAC8
SCHEMBL20344747 0.78 BRD4 (0.42) BRD4CREBBPHDAC1HDAC8HDAC6
SCHEMBL20344739 0.78 BRD4 (0.42) IDH1BRD4CREBBPHDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3342766-A1 SMALL MOLECULE COMPOUND FOR ENHANCING PLANT STRESS RESISTANCE Shanghai Institutes for Biological Sciences, Chinese Academy of Sciences (CN) 2018-07-04 EP disclosed