SCHEMBL20360950

SCHEMBL20360950

C[C@H](CCO)Cc1ccc(Br)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.39
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
TRPA1 O75762 1/20 0.34
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GRM2 Q14416 1/20 0.32
ADRA2A P08913 2/20 0.32
ADRA2B P18089 2/20 0.32
ADRA2C P18825 2/20 0.32
PLAU P00749 1/20 0.32
MBOAT4 Q96T53 1/20 0.32
RAB9A P51151 5/20 0.31
SIRT2 Q8IXJ6 1/20 0.31
FDPS P14324 1/20 0.31
MAPT P10636 2/20 0.31
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
TP53 P04637 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27859444 1.00 GBA1 (0.39) GBA1ESR1ESR2TRPA1ALDH1A1
SCHEMBL5144435 0.79 GBA1 (0.43) GBA1ESR1ESR2ALDH1A1KDM4E
SCHEMBL30305975 0.79 GBA1 (0.43) GBA1ESR1ESR2ALDH1A1KDM4E
SCHEMBL14464977 0.79 GBA1 (0.43) GBA1ESR1ESR2ALDH1A1KDM4E
SCHEMBL5344274 0.78 GBA1 (0.46) GBA1ESR1ESR2ALDH1A1KDM4E
SCHEMBL14321841 0.77 GBA1 (0.39) GBA1ESR1ESR2ALDH1A1KDM4E
SCHEMBL20361529 0.77 GBA1 (0.39) GBA1ESR1ESR2ALDH1A1KDM4E
SCHEMBL23158732 0.74 GBA1 (0.41) GBA1ESR1ESR2ALDH1A1KDM4E
SCHEMBL5728691 0.73 ACACB (0.41) TRPA1RAB9AKMT2AMEN1NPC1
SCHEMBL13643094 0.73 ACACB (0.41) TRPA1RAB9AKMT2AMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3565809-A1 PYRIDIN-3-YL ACETIC ACID DERIVATIVES AS INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION ViiV Healthcare UK (No.5) Limited (GB) 2019-11-13 EP disclosed
WO-2018127800-A1 PYRIDIN-3-YL ACETIC ACID DERIVATIVES AS INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV Healthcare UK (No.5) Limited (GB) 2018-07-12 WO disclosed