SCHEMBL20375005

SCHEMBL20375005

Cc1cnc2[nH]cc(C(=O)c3c(O)ccc(N)c3F)c2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 9/20 0.53
CYP2C19 P33261 7/20 0.52
CYP3A4 P08684 4/20 0.50
RIPK2 O43353 2/20 0.41
RAF1 P04049 2/20 0.41
KDR P35968 2/20 0.41
MAP2K2 P36507 2/20 0.41
TGFBR2 P37173 2/20 0.41
NEK2 P51955 2/20 0.41
MAP2K1 Q02750 2/20 0.41
TNK2 Q07912 2/20 0.41
MAP2K5 Q13163 2/20 0.41
PTK6 Q13882 2/20 0.41
NEK11 Q8NG66 2/20 0.41
MAP3K20 Q9NYL2 2/20 0.41
MAP4K5 Q9Y4K4 2/20 0.41
BMPR1B O00238 1/20 0.41
PLK4 O00444 1/20 0.41
PIR O00625 1/20 0.41
AURKA O14965 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL293715 0.90 BRAF (0.64) BRAFCYP2C19CYP3A4RIPK2RAF1
SCHEMBL17145187 0.90 BRAF (0.54) BRAFCYP2C19CYP3A4RIPK2RAF1
SCHEMBL19068717 0.87 BRAF (0.41) BRAFCYP2C19CYP3A4RIPK2RAF1
SCHEMBL19068718 0.87 CYP2C19 (0.41) BRAFCYP2C19CYP3A4RIPK2RAF1
SCHEMBL20375065 0.87 BRAF (0.48) BRAFCYP2C19CYP3A4RIPK2RAF1
SCHEMBL3705469 0.82 CYP3A4 (0.52) BRAFCYP2C19CYP3A4RIPK2RAF1
SCHEMBL15600583 0.81 BRAF (0.49) BRAFCYP3A4KDRNEK2MAP2K1
SCHEMBL10262647 0.80 BRAF (0.58) BRAFCYP2C19CYP3A4RIPK2RAF1
SCHEMBL19413965 0.80 BRAF (0.57) BRAFCYP2C19CYP3A4RIPK2RAF1
SCHEMBL3703309 0.80 BRAF (0.51) BRAFCYP2C19CYP3A4RIPK2RAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2861591-B1 SYNTHESIS OF PYRROLO[2,3-B]PYRIDINES PLEXXIKON INC (US) 2018-07-11 EP disclosed