SCHEMBL20458440

SCHEMBL20458440

CCCCC(=O)N1CCN(c2nc(C3CC3)c(Oc3ccnc(Cl)c3)cc2C#N)CC1C

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 17/20 0.43
PIK3CD O00329 1/20 0.40
PIK3R1 P27986 1/20 0.40
CHRM1 P11229 1/20 0.38
GRM1 Q13255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15901365 0.93 IDH1 (0.44) IDH1PIK3CDPIK3R1GRM1
SCHEMBL14249966 0.93 IDH1 (0.44) IDH1PIK3CDPIK3R1GRM1
SCHEMBL14250795 0.91 IDH1 (0.52) IDH1
SCHEMBL15900889 0.91 IDH1 (0.52) IDH1
SCHEMBL17996938 0.85 MAP4K4 (0.39) IDH1GRM1
SCHEMBL14250205 0.84 IDH1 (0.49) IDH1
SCHEMBL14315319 0.84 IDH1 (0.49) IDH1
SCHEMBL14250336 0.83 IDH1 (0.52) IDH1
SCHEMBL14250335 0.83 IDH1 (0.52) IDH1
SCHEMBL14315350 0.82 IDH1 (0.35) IDH1PIK3CDPIK3R1GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2721019-B1 THERAPEUTICALLY ACTIVE COMPOSITIONS AND THEIR METHODS OF USE AGIOS PHARMACEUTICALS INC (US) 2018-08-08 EP disclosed