SCHEMBL20490502

SCHEMBL20490502

O=C(NO)C(c1ccccc1)c1ccc(-c2csc3ccccc23)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 10/20 0.55
HDAC7 Q8WUI4 5/20 0.55
HDAC5 Q9UQL6 5/20 0.55
HDAC2 Q92769 4/20 0.55
HDAC3 O15379 3/20 0.55
HDAC1 Q13547 3/20 0.55
HDAC10 Q969S8 3/20 0.55
HDAC11 Q96DB2 3/20 0.55
HDAC8 Q9BY41 3/20 0.55
HDAC6 Q9UBN7 3/20 0.55
HDAC9 Q9UKV0 3/20 0.55
APP P05067 2/20 0.47
ERN1 O75460 2/20 0.43
NPC1 O15118 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
CTSD P07339 1/20 0.40
POLB P06746 1/20 0.39
CYP2C9 P11712 1/20 0.39
CSNK1D P48730 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20490230 0.89 HDAC4 (0.51) HDAC4HDAC7HDAC5HDAC2HDAC3
SCHEMBL20490126 0.78 HDAC3 (0.57) HDAC4HDAC7HDAC5HDAC2HDAC3
SCHEMBL2839404 0.77 HDAC4 (0.60) HDAC4HDAC7HDAC5HDAC2HDAC3
SCHEMBL2842461 0.76 HDAC4 (0.81) HDAC4HDAC7HDAC5HDAC2HDAC3
SCHEMBL20490165 0.76 HDAC4 (0.58) HDAC4HDAC7HDAC5HDAC2HDAC3
SCHEMBL20490498 0.76 HDAC4 (0.58) HDAC4HDAC7HDAC5HDAC2HDAC3
SCHEMBL2839032 0.74 HDAC4 (1.00) HDAC4HDAC7HDAC5HDAC2HDAC3
SCHEMBL20490215 0.73 HDAC4 (0.64) HDAC4HDAC7HDAC5HDAC2HDAC3
SCHEMBL20490457 0.73 HDAC4 (0.64) HDAC4HDAC7HDAC5HDAC2HDAC3
SCHEMBL5766614 0.73 ERN1 (0.51) HDAC2APPERN1NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139850-B1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC (CA) 2018-09-12 EP claimed
EP-2139850-B1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC (CA) 2018-09-12 EP disclosed
CN-101679220-A Histone deacetylase inhibitor METHYLGENE INC 2010-03-24 CN disclosed