SCHEMBL20523716

SCHEMBL20523716

Fc1ccc(CC(F)(F)F)cc1Br

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
KDM4E B2RXH2 3/20 0.45
PARP1 P09874 2/20 0.36
FAAH O00519 1/20 0.34
VCP P55072 1/20 0.33
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
MAOB P27338 2/20 0.32
PTPN7 P35236 1/20 0.32
DUSP3 P51452 1/20 0.32
MAOA P21397 1/20 0.32
KDR P35968 1/20 0.32
GRIN1 Q05586 1/20 0.31
GRIN2B Q13224 1/20 0.31
IDO1 P14902 1/20 0.30
TDO2 P48775 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18097710 0.83 KDM1A (0.35) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1
SCHEMBL13905164 0.82 CYP1A2 (0.47) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1
SCHEMBL7107363 0.78 CA12 (0.38) KDM4EALDH1A1TSHR
SCHEMBL23629171 0.78 HPGD (0.35) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1
SCHEMBL30986323 0.78 HPGD (0.35) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1
SCHEMBL29418197 0.76 CYP1A2 (0.53) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1
SCHEMBL20523441 0.76
SCHEMBL333551 0.76 CYP1A2 (0.53) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1
SCHEMBL11244115 0.76 KDM4E (0.49) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1
SCHEMBL2657319 0.75 CYP1A2 (0.53) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023114823-A1 BENZOTHIOPHENE DERIVATIVES AS RXFP1 AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2023-06-22 WO disclosed
WO-2023077070-A1 RXFP1 AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2023-05-04 WO disclosed
WO-2018183601-A1 MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO DOW AGROSCIENCES LLC (US) 2018-10-04 WO disclosed