SCHEMBL2053552

SCHEMBL2053552

N[C@@]1(C(=O)O)CC[C@@H](c2ccc(Br)cc2)C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 6/20 0.45
CYP2C19 P33261 3/20 0.45
GRM2 Q14416 2/20 0.45
GRM3 Q14832 2/20 0.45
CYP1A2 P05177 2/20 0.45
TDP1 Q9NUW8 2/20 0.45
GRM8 O00222 2/20 0.45
GRM6 O15303 2/20 0.45
ALOX15 P16050 1/20 0.45
LMNA P02545 1/20 0.45
GRM5 P41594 1/20 0.45
MTOR P42345 1/20 0.45
GRM1 Q13255 1/20 0.45
PLCB1 Q9NQ66 1/20 0.45
TSHR P16473 1/20 0.45
KDM1A O60341 4/20 0.39
RCOR1 Q9UKL0 4/20 0.39
ESR2 Q92731 4/20 0.37
ESR1 P03372 1/20 0.37
LIG1 P18858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15953786 1.00 GRM4 (0.45) GRM4CYP2C19GRM2GRM3CYP1A2
SCHEMBL2053441 1.00 GRM4 (0.45) GRM4CYP2C19GRM2GRM3CYP1A2
SCHEMBL15953683 1.00 GRM4 (0.45) GRM4CYP2C19GRM2GRM3CYP1A2
SCHEMBL2313610 1.00 GRM4 (0.45) GRM4CYP2C19GRM2GRM3CYP1A2
SCHEMBL2313607 1.00 GRM4 (0.45) GRM4CYP2C19GRM2GRM3CYP1A2
SCHEMBL2041074 1.00 GRM4 (0.45) GRM4CYP2C19GRM2GRM3CYP1A2
SCHEMBL2042819 1.00 GRM4 (0.45) GRM4CYP2C19GRM2GRM3CYP1A2
Hydrochloric Acid SCHEMBL28474763 0.98 GRM4 (0.44) GRM4CYP2C19GRM2GRM3CYP1A2
SCHEMBL14140688 0.88 ESR2 (0.37) KDM1ARCOR1ESR2ESR1LIG1
SCHEMBL10299842 0.86 KDM1A (0.39) LMNATSHRKDM1ARCOR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7956195-B2 reacting arylboronic acids with a cycloalkanone, in the presence of a rhodium catalyst or BINAP, to form a substituted arylcycloalkanone, then formin of a hydantoin, alkylation of the hydantoin, resolution, hydrolysis of the hydantoin to the amino acids and esterification of acids; chemical intermediates ABBOTT LABORATORIES (US) 2011-06-07 US disclosed