SCHEMBL20544273

SCHEMBL20544273

CCc1c(C)c(Cc2ccc(F)c(C(=O)N3CCCNCC3)c2)n[nH]c1=O

nearest known ligand 0.73

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 20/20 0.73
PARP3 Q9Y6F1 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL3912532 0.95 PARP1 (0.67) PARP1PARP3
SCHEMBL20544379 0.94 PARP1 (0.72) PARP1PARP3
SCHEMBL20544232 0.94 PARP1 (0.74) PARP1PARP3
SCHEMBL20544383 0.92 PARP1 (0.77) PARP1PARP3
Trifluoroacetic Acid SCHEMBL3910680 0.89 PARP1 (0.66) PARP1PARP3
Trifluoroacetic Acid SCHEMBL3912153 0.89 PARP1 (0.68) PARP1PARP3
SCHEMBL4248757 0.88 PARP1 (0.63) PARP1
SCHEMBL17160852 0.88 PARP1 (0.78) PARP1PARP3
SCHEMBL20544655 0.88 PARP1 (0.71) PARP1PARP3
Trifluoroacetic Acid SCHEMBL3911477 0.87 PARP1 (0.70) PARP1PARP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029551-B1 PYRIDINONE AND PYRIDAZINONE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) MSD ITALIA SRL (IT) 2018-10-31 EP claimed