SCHEMBL20544385

SCHEMBL20544385

Cc1c(Cc2ccc(F)c(N3C(=O)NC(C)C3=O)c2)n[nH]c(=O)c1C

nearest known ligand 0.55

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 20/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4244380 0.92 PARP1 (0.49) PARP1
SCHEMBL8050461 0.85 PARP1 (0.74) PARP1
SCHEMBL2208157 0.85 PARP1 (0.74) PARP1
SCHEMBL8242343 0.85 PARP1 (0.67) PARP1
SCHEMBL1806111 0.85 PARP1 (0.67) PARP1
SCHEMBL8055652 0.85 PARP1 (0.74) PARP1
SCHEMBL5131450 0.81 PARP1 (0.79) PARP1
SCHEMBL1804463 0.73 PARP1 (0.47) PARP1
SCHEMBL3076203 0.71 PARP1 (0.67) PARP1
SCHEMBL3068304 0.71 PARP1 (0.49) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029551-B1 PYRIDINONE AND PYRIDAZINONE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) MSD ITALIA SRL (IT) 2018-10-31 EP claimed