SCHEMBL20548965

SCHEMBL20548965

[CH2]CN1CCc2nc(Nc3ncc(F)c(-c4cc(F)c5nc(C)n(C(C)C)c5c4)n3)ccc2C1

nearest known ligand 0.87

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.87
CDK1 P06493 11/20 0.87
CCNB1 P14635 7/20 0.87
CCNE1 P24864 7/20 0.87
CDK2 P24941 16/20 0.85
CDK6 Q00534 16/20 0.85
CDK7 P50613 6/20 0.84
CDK9 P50750 6/20 0.84
CDK5 Q00535 3/20 0.81
CHEK1 O14757 1/20 0.81
CCNT1 O60563 1/20 0.81
JAK2 O60674 1/20 0.81
CHEK2 O96017 1/20 0.81
EGFR P00533 1/20 0.81
RAF1 P04049 1/20 0.81
NTRK1 P04629 1/20 0.81
PDGFRB P09619 1/20 0.81
SRC P12931 1/20 0.81
BRAF P15056 1/20 0.81
PDGFRA P16234 1/20 0.81

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17477262 0.93 CDK4 (1.00) CDK4CDK1CCNB1CCNE1CDK2
SCHEMBL18288930 0.92 CDK4 (0.89) CDK4CDK1CCNB1CCNE1CDK2
SCHEMBL17485310 0.92 CDK4 (1.00) CDK4CDK1CCNB1CCNE1CDK2
SCHEMBL19089098 0.92 CDK4 (0.91) CDK4CDK1CCNB1CCNE1CDK2
SCHEMBL22280579 0.91 CDK4 (0.85) CDK4CDK1CCNB1CCNE1CDK2
Hydrochloric Acid SCHEMBL20548753 0.91 CDK4 (0.90) CDK4CDK1CCNB1CCNE1CDK2
SCHEMBL18288922 0.91 CDK4 (1.00) CDK4CDK1CCNB1CCNE1CDK2
SCHEMBL18288771 0.91 CDK4 (1.00) CDK4CDK1CCNB1CCNE1CDK2
SCHEMBL19088970 0.91 CDK4 (1.00) CDK4CDK1CCNB1CCNE1CDK2
SCHEMBL19089044 0.91 CDK4 (0.86) CDK4CDK1CCNB1CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3398947-A1 NITROGEN-CONTAINING FUSED HETEROCYCLIC COMPOUND, AS WELL AS PREPARATION METHOD, INTERMEDIATE, COMPOSITION AND APPLICATION THEREOF Shanghai Pharmaceuticals Holding Co., Ltd. (CN) 2018-11-07 EP disclosed