SCHEMBL20558294

SCHEMBL20558294

CCOC(=O)c1cccc2c1CN(C(=O)OC(C)(C)C)CC2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.51
ESR2 Q92731 1/20 0.48
NR1H2 P55055 1/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
TMEM97 Q5BJF2 2/20 0.45
SIGMAR1 Q99720 2/20 0.45
MAPK1 P28482 1/20 0.45
TP53 P04637 1/20 0.44
POLB P06746 1/20 0.44
F12 P00748 1/20 0.43
PRMT5 O14744 2/20 0.42
WDR77 Q9BQA1 2/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ABHD6 Q9BV23 1/20 0.42
DDB1 Q16531 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30670170 1.00 ADORA1 (0.51) ADORA1ESR2NR1H2MEN1KMT2A
SCHEMBL21496681 0.90 DDB1 (0.48) ADORA1ESR2MEN1KMT2AMAPK1
SCHEMBL19739032 0.87 ESR2 (0.51) ESR2NR1H2TMEM97SIGMAR1MAPK1
SCHEMBL1570606 0.86 ESR2 (0.54) ADORA1ESR2NR1H2TMEM97SIGMAR1
SCHEMBL29801280 0.86 ESR2 (0.54) ADORA1ESR2NR1H2TMEM97SIGMAR1
SCHEMBL14895889 0.84 ESR2 (0.53) ESR2NR1H2TMEM97SIGMAR1MAPK1
SCHEMBL24628746 0.83 ESR2 (0.56) ADORA1ESR2NR1H2MEN1KMT2A
SCHEMBL19608875 0.83 ESR2 (0.56) ESR2NR1H2TMEM97SIGMAR1MAPK1
SCHEMBL25107642 0.82 ESR2 (0.51) ADORA1ESR2NR1H2TMEM97SIGMAR1
SCHEMBL14868188 0.81 ESR2 (0.50) ESR2NR1H2TMEM97SIGMAR1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116783160-A Libraries of compounds 中外制药株式会社 2023-09-19 CN disclosed
WO-2018205948-A1 COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-11-15 WO disclosed