SCHEMBL20568595

SCHEMBL20568595

COC(=O)n1cc(I)c(C)c1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
P2RX4 Q99571 2/20 0.37
HTT P42858 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA3 P34903 1/20 0.36
ABCB1 P08183 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
LPO P22079 1/20 0.35
GRM6 O15303 1/20 0.35
GRM5 P41594 1/20 0.35
RAB9A P51151 2/20 0.34
MAPT P10636 2/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP3A4 P08684 2/20 0.34
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7209262 0.74 KMT2A (0.47) BCHEMEN1KMT2AHTTGABRA1
SCHEMBL20569871 0.73 BCHE (0.39) BCHEMEN1KMT2AP2RX4HTT
SCHEMBL1127344 0.70 MEN1 (0.42) BCHEMEN1KMT2AHTTLPO
Biphenyl SCHEMBL3255863 0.61 TSHR (0.54) KMT2ARAB9AMAPTALDH1A1SMN1; SMN2
SCHEMBL9791225 0.61 KMT2A (0.60) MEN1KMT2AHTTRAB9AMAPT
SCHEMBL8076273 0.61 KMT2A (0.67) MEN1KMT2ARAB9AMAPTALDH1A1
SCHEMBL10959666 0.61 GRM5 (0.57) MEN1KMT2AGABRA1GABRG2GABRB3
Biphenyl SCHEMBL27677322 0.60 TSHR (0.52) KMT2ARAB9AMAPTALDH1A1SMN1; SMN2
Biphenyl SCHEMBL27819830 0.60 SMN1; SMN2 (0.56) KMT2ARAB9AMAPTALDH1A1SMN1; SMN2
Biphenyl SCHEMBL27492413 0.60 TSHR (0.52) KMT2ARAB9AMAPTALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3630728-A1 INHIBITORS OF METALLO-BETA-LACTAMASES Oxford University Innovation Limited (GB) 2020-04-08 EP disclosed
WO-2018215799-A1 INHIBITORS OF METALLO-BETA-LACTAMASES OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2018-11-29 WO disclosed