SCHEMBL20568944

SCHEMBL20568944

CC(C)(C)OC(=O)N1CCc2cc(C#Cc3ccc(CO)cc3)ccc2C1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 2/20 0.61
NR1H2 P55055 1/20 0.54
GPR119 Q8TDV5 1/20 0.41
MAPK1 P28482 1/20 0.41
ACACB O00763 1/20 0.40
MAPT P10636 1/20 0.40
ABHD6 Q9BV23 2/20 0.40
HDAC1 Q13547 1/20 0.40
TMEM97 Q5BJF2 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
DDB1 Q16531 1/20 0.39
CRBN Q96SW2 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
ESR1 P03372 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
NAMPT P43490 2/20 0.38
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL168265 0.87 ESR2 (0.70) ESR2NR1H2GPR119MAPK1MAPT
SCHEMBL29407529 0.87 ESR2 (0.70) ESR2NR1H2GPR119MAPK1MAPT
SCHEMBL29407557 0.83 NR1H2 (0.69) ESR2NR1H2GPR119MAPK1MAPT
SCHEMBL1285596 0.83 NR1H2 (0.69) ESR2NR1H2GPR119MAPK1MAPT
SCHEMBL3011371 0.82 ESR2 (0.63) ESR2NR1H2MAPK1MAPTABHD6
SCHEMBL3009208 0.82 ESR2 (0.69) ESR2NR1H2MAPK1MAPTABHD6
SCHEMBL30548176 0.82 ESR2 (0.69) ESR2NR1H2GPR119MAPK1MAPT
SCHEMBL451998 0.82 ESR2 (0.69) ESR2NR1H2GPR119MAPK1MAPT
SCHEMBL30409090 0.82 ESR2 (0.69) ESR2NR1H2MAPK1MAPTABHD6
SCHEMBL1365302 0.81 ESR2 (0.67) ESR2NR1H2MAPK1MAPTABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018216823-A1 ALPHA-AMINO AMIDE DERIVATIVES TAISHO PHARMACEUTICAL CO., LTD. (JP) 2018-11-29 WO disclosed