SCHEMBL20577115

SCHEMBL20577115

CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(Cc4ccccc4)CC3)cc21

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 1/20 0.73
KDM4E B2RXH2 8/20 0.70
ALDH1A1 P00352 5/20 0.70
HPGD P15428 5/20 0.70
MEN1 O00255 5/20 0.70
KMT2A Q03164 5/20 0.70
HTT P42858 4/20 0.70
HSD17B10 Q99714 3/20 0.70
LMNA P02545 2/20 0.70
TSHR P16473 2/20 0.70
USP2 O75604 1/20 0.70
SMN1; SMN2 Q16637 1/20 0.70
BRD4 O60885 1/20 0.69
CYP2J2 P51589 1/20 0.69
NPSR1 Q6W5P4 1/20 0.69
NPC1 O15118 1/20 0.67
MAPT P10636 1/20 0.67
PIK3CG P48736 3/20 0.65
PIK3CD O00329 2/20 0.64
PIK3R1 P27986 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30306107 1.00 DRD3 (0.73) DRD3KDM4EALDH1A1HPGDMEN1
Hydrochloric Acid SCHEMBL25379465 0.99 DRD3 (0.72) DRD3KDM4EALDH1A1HPGDMEN1
Hydrochloric Acid SCHEMBL30306094 0.99 DRD3 (0.72) DRD3KDM4EALDH1A1HPGDMEN1
SCHEMBL25379277 0.94 DRD3 (0.68) DRD3KDM4EALDH1A1HPGDMEN1
SCHEMBL30306127 0.94 DRD3 (0.68) DRD3KDM4EALDH1A1HPGDMEN1
Hydrochloric Acid SCHEMBL25379605 0.94 DRD3 (0.67) DRD3KDM4EALDH1A1HPGDMEN1
Hydrochloric Acid SCHEMBL31679577 0.94 DRD3 (0.67) DRD3KDM4EALDH1A1HPGDMEN1
SCHEMBL26193832 0.93 DRD3 (0.72) DRD3KDM4EALDH1A1HPGDMEN1
SCHEMBL25380525 0.93 DRD3 (0.71) DRD3KDM4EALDH1A1HPGDMEN1
SCHEMBL30306102 0.93 DRD3 (0.71) DRD3KDM4EALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3630779-B1 ANTIBIOTIC RESISTANCE BREAKERS KING S COLLEGE LONDON (GB) 2025-09-03 EP disclosed
US-11746116-B2 Antibiotic resistance breakers KING'S COLLEGE LONDON (GB) 2023-09-05 US disclosed
US-11746116-B2 Antibiotic resistance breakers KING'S COLLEGE LONDON (GB) 2023-09-05 US disclosed
US-11746116-B2 Antibiotic resistance breakers KING'S COLLEGE LONDON (GB) 2023-09-05 US disclosed
CN-110869373-B Antibiotic resistance disruptors 伦敦皇家学院 2023-03-07 CN disclosed
EP-3630779-A1 ANTIBIOTIC RESISTANCE BREAKERS Kings College London (GB) 2020-04-08 EP disclosed
CN-110869373-A Antibiotic resistance disruptors 伦敦皇家学院 2020-03-06 CN disclosed
WO-2018220365-A1 ANTIBIOTIC RESISTANCE BREAKERS KING'S COLLEGE LONDON (GB) 2018-12-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11746116-B2 Antibiotic resistance breakers ABCC1, ARL1, AKR1C3 DRD3 594/4885KDM4E 3599/4885ALDH1A1 481/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.