SCHEMBL20613019

SCHEMBL20613019

CC(O)(Cn1cncn1)c1ccc(Oc2ccccc2)nc1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.43
CYP3A4 P08684 6/20 0.38
CYP2C9 P11712 5/20 0.38
CYP2C19 P33261 5/20 0.38
CYP19A1 P11511 2/20 0.38
LMNA P02545 2/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
ADRA1A P35348 1/20 0.38
CYP51A1 Q16850 1/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 2/20 0.38
TSHR P16473 1/20 0.37
AR P10275 1/20 0.36
ALOX15 P16050 1/20 0.34
KMT2A Q03164 2/20 0.33
CYP2B6 P20813 1/20 0.33
CYP3A5 P20815 1/20 0.33
CYP3A7 P24462 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20597452 0.91 CYP3A4 (0.38) HSP90AA1CYP3A4CYP2C9CYP2C19CYP19A1
SCHEMBL20597246 0.91 CYP3A4 (0.38) HSP90AA1CYP3A4CYP2C9CYP2C19CYP19A1
SCHEMBL20597170 0.91 CYP3A4 (0.38) HSP90AA1CYP3A4CYP2C9CYP2C19CYP19A1
SCHEMBL20537234 0.90 CYP3A4 (0.44) HSP90AA1CYP3A4CYP2C9CYP2C19CYP19A1
SCHEMBL20537212 0.90 CYP3A4 (0.44) HSP90AA1CYP3A4CYP2C9CYP2C19CYP19A1
SCHEMBL18542630 0.90 CYP3A4 (0.44) HSP90AA1CYP3A4CYP2C9CYP2C19CYP19A1
SCHEMBL20537217 0.90 CYP3A4 (0.37) HSP90AA1CYP3A4CYP2C9CYP2C19CYP19A1
SCHEMBL20537209 0.90 CYP3A4 (0.37) HSP90AA1CYP3A4CYP2C9CYP2C19CYP19A1
SCHEMBL29354915 0.90 CYP3A4 (0.37) HSP90AA1CYP3A4CYP2C9CYP2C19CYP19A1
SCHEMBL20471552 0.90 CYP3A4 (0.37) HSP90AA1CYP3A4CYP2C9CYP2C19CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3421460-A1 2-[(4-ALKYLPHENOXY)-PYRIDINYL]-1-(1,2,4-TRIAZOL-1-YL)ALKAN-2-OL FUNGICIDES Bayer Aktiengesellschaft (DE) 2019-01-02 EP disclosed