SCHEMBL20616645

SCHEMBL20616645

C/C=C1\CCN(C(=O)OCC)CC1(C)C

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 12/20 0.54
TSHR P16473 1/20 0.39
POLB P06746 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPT P10636 2/20 0.37
ABL1 P00519 1/20 0.37
RIN1 Q13671 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GAA P10253 2/20 0.36
RECQL P46063 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29915315 0.83 GRM5 (0.58) GRM5CYP3A4
SCHEMBL6308517 0.80 GRM5 (0.48) GRM5TSHRPOLBALDH1A1HTT
SCHEMBL29915494 0.79 GRM5 (0.66) GRM5CYP3A4
SCHEMBL13901291 0.78 GRM5 (0.35) GRM5LMNA
SCHEMBL3126731 0.77 GRM5 (0.45) GRM5SMN1; SMN2
SCHEMBL20658743 0.77 GRM5 (0.45) GRM5SMN1; SMN2
SCHEMBL3126738 0.77 GRM5 (0.45) GRM5SMN1; SMN2
SCHEMBL3126917 0.77 GRM5 (0.44) GRM5ALDH1A1RECQLKDM4ELMNA
SCHEMBL3126909 0.77 GRM5 (0.44) GRM5ALDH1A1RECQLKDM4ELMNA
SCHEMBL22619524 0.75 GRM5 (0.78) GRM5CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019002571-A1 HETEROCYCLYLMETHYLIDENE DERIVATIVES AND THEIR USE AS MODULATORS OF mGluR5 RECEPTORS RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA SPA (IT) 2019-01-03 WO disclosed