SCHEMBL20649155

SCHEMBL20649155

CCn1nc(C(=O)NC2NC(C)=CS2)c2c1-c1nc(N)ncc1CC2(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 19/20 0.37
CCNA2 P20248 5/20 0.37
CDK4 P11802 4/20 0.37
CCND3 P30281 3/20 0.37
CDK6 Q00534 3/20 0.37
AURKA O14965 14/20 0.36
GAK O14976 1/20 0.35
BUB1 O43683 1/20 0.35
CCNT1 O60563 1/20 0.35
ULK1 O75385 1/20 0.35
STK16 O75716 1/20 0.35
PRKD3 O94806 1/20 0.35
LATS1 O95835 1/20 0.35
ABL1 P00519 1/20 0.35
EGFR P00533 1/20 0.35
NTRK1 P04629 1/20 0.35
LCK P06239 1/20 0.35
FYN P06241 1/20 0.35
CDK1 P06493 1/20 0.35
YES1 P07947 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20648965 0.92 CDK2 (0.38) CDK2CCNA2CDK4CCND3CDK6
SCHEMBL20649323 0.92 CDK2 (0.37) CDK2CCNA2CDK4CCND3CDK6
SCHEMBL20649300 0.85 CDK2 (0.36) CDK2CCNA2CDK4CCND3CDK6
SCHEMBL20648930 0.81 CDK4 (0.30) CDK2CCNA2CDK4CCND3CDK6
SCHEMBL20649144 0.78 CDK2 (0.46) CDK2CCNA2CDK4CCND3CDK6
SCHEMBL30183501 0.78 GCK (0.39) CDK2CCNA2CDK4CCND3CDK6
SCHEMBL20649154 0.78 GCK (0.39) CDK2CCNA2CDK4CCND3CDK6
SCHEMBL20649094 0.74
SCHEMBL20649409 0.71 CDK2 (0.36) CDK2CCNA2CDK4CCND3CDK6
SCHEMBL30183884 0.71 CDK2 (0.36) CDK2CCNA2CDK4CCND3CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019011715-A1 PYRAZOLO-QUINAZOLINE DERIVATIVES AS CHOLINE KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2019-01-17 WO disclosed