SCHEMBL2065

SCHEMBL2065

COC(=O)[C@H](Cc1ccc(F)cc1)NCc1ccc(-c2ccccc2C#N)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
ITGB1 P05556 4/20 0.48
ITGA4 P13612 4/20 0.48
PTPN1 P18031 1/20 0.47
MME P08473 1/20 0.45
MYC P01106 1/20 0.44
WDR5 P61964 1/20 0.44
ACHE P22303 1/20 0.43
NOS2 P35228 3/20 0.43
NOS3 P29474 2/20 0.43
NOS1 P29475 2/20 0.43
FFAR1 O14842 1/20 0.43
AKR1B1 P15121 1/20 0.43
ITGB7 P26010 3/20 0.42
ATM Q13315 2/20 0.41
ESR2 Q92731 1/20 0.41
ANPEP P15144 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2693 0.86 ITGB1 (0.46) ITGB1ITGA4PTPN1MMEMYC
SCHEMBL2772 0.84 ITGB1 (0.44) ITGB1ITGA4PTPN1MMEMYC
SCHEMBL2132 0.81 MYC (0.47) ITGB1ITGA4PTPN1MMEMYC
SCHEMBL2870 0.81 MYC (0.47) ITGB1ITGA4PTPN1MMEMYC
SCHEMBL2174 0.79 MYC (0.45) CA12CA7CA9CA14ITGB1
SCHEMBL2432 0.79 MYC (0.45) CA12CA7CA9CA14ITGB1
SCHEMBL8065614 0.79 MYC (0.45) CA12CA7CA9CA14ITGB1
Hydrochloric Acid SCHEMBL3526296 0.78 MYC (0.45) CA12CA7CA9CA14ITGB1
Hydrochloric Acid SCHEMBL15663201 0.78 MYC (0.45) CA12CA7CA9CA14ITGB1
SCHEMBL7177998 0.78 MME (0.52) ITGB1ITGA4PTPN1MMEMYC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965592-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1999-10-12 US disclosed
EP-0443983-B1 Acyl compounds CIBA GEIGY AG (CH) 1996-02-28 EP disclosed
US-5399578-A Hypotensive; valsartan; high blood pressure and cardiac insufficiency CIBA-GEIGY CORP (US) 1995-03-21 US disclosed
EP-0443983-A1 Acyl compounds CIBA-GEIGY AG (CH) 1991-08-28 EP disclosed