SCHEMBL20669783

SCHEMBL20669783

CC(=O)c1c(C)c(C)nc2ccccc12

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.77
HSD17B10 Q99714 2/20 0.68
TP53 P04637 1/20 0.68
HTT P42858 3/20 0.57
KMT2A Q03164 4/20 0.54
MEN1 O00255 3/20 0.54
TSHR P16473 1/20 0.53
ALDH1A1 P00352 3/20 0.50
DHODH Q02127 2/20 0.50
GPR3 P46089 1/20 0.50
GAA P10253 1/20 0.50
MAPT P10636 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
CYP1A2 P05177 1/20 0.50
HPGD P15428 1/20 0.50
NUDT1 P36639 1/20 0.50
KDM4E B2RXH2 1/20 0.50
SMN1; SMN2 Q16637 3/20 0.48
ERN1 O75460 1/20 0.46
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13957825 0.87 PDE10A (1.00) PDE10AHSD17B10TP53HTTKMT2A
SCHEMBL15487702 0.84 HSD17B10 (0.66) PDE10AHSD17B10TP53HTTKMT2A
SCHEMBL20659212 0.84 PDE10A (0.75) PDE10AHSD17B10TP53HTTKMT2A
SCHEMBL29864783 0.84 PDE10A (0.75) PDE10AHSD17B10TP53HTTKMT2A
SCHEMBL29952587 0.84 HSD17B10 (0.71) PDE10AHSD17B10TP53HTTKMT2A
SCHEMBL20669707 0.84 PDE10A (0.75) PDE10AHSD17B10TP53HTTKMT2A
SCHEMBL20669570 0.84 PDE10A (0.75) PDE10AHSD17B10TP53HTTKMT2A
SCHEMBL12220557 0.83 HSD17B10 (0.62) PDE10AHSD17B10TP53HTTKMT2A
SCHEMBL21878637 0.81 MEN1 (0.75) PDE10AHSD17B10TP53HTTKMT2A
SCHEMBL6654332 0.81 HSD17B10 (1.00) PDE10AHSD17B10TP53HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019016269-A1 AMINE OR (THIO)AMIDE CONTAINING LXR MODULATORS PHENEX-FXR GMBH (DE) 2019-01-24 WO disclosed