SCHEMBL20689593

SCHEMBL20689593

CC(C)n1cc(Br)c2cccnc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 2/20 0.45
SLC22A12 Q96S37 1/20 0.42
PDE4A P27815 3/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
RET P07949 2/20 0.38
KDR P35968 2/20 0.38
TYK2 P29597 1/20 0.37
AXL P30530 1/20 0.37
GSK3B P49841 2/20 0.35
KCNH2 Q12809 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 2/20 0.35
HSP90AA1 P07900 2/20 0.35
APAF1 O14727 1/20 0.35
TDP2 O95551 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12889428 0.80 PDE4A (0.42) ELANEPDE4APDE4BPDE4CPDE4D
SCHEMBL27681105 0.79 ELANE (0.43) ELANESLC22A12PDE4AAXLKCNH2
SCHEMBL27251595 0.79 PSMB5 (0.44) PDE4APDE4BPDE4CPDE4DMEN1
SCHEMBL12874831 0.79 PDE4A (0.41) ELANEPDE4APDE4BPDE4CPDE4D
SCHEMBL26628372 0.79 RET (0.43) PDE4APDE4BPDE4CPDE4DRET
SCHEMBL31725474 0.79 RET (0.43) PDE4APDE4BPDE4CPDE4DRET
SCHEMBL26354834 0.79 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DRET
SCHEMBL414164 0.78 ELANE (0.42) ELANESLC22A12PDE4AAXLKCNH2
SCHEMBL1892910 0.78 DYRK1A (0.49) ELANESLC22A12AXLGSK3BMEN1
SCHEMBL30731192 0.78 DYRK1A (0.49) ELANESLC22A12AXLGSK3BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022257568-A1 AZAINDOLE PYRIMIDINAMINE HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 中国药科大学 2022-12-15 WO disclosed
WO-2019023468-A1 TYK2 INHIBITORS AND USES THEREOF NIMBUS LAKSHMI, INC. (US) 2019-01-31 WO disclosed