SCHEMBL20698299

SCHEMBL20698299

COc1cc(F)c(-c2c(C)nn(C)c2N(N)c2c(N)cc(Cl)cc2F)c(F)c1

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.37
PDE10A Q9Y233 1/20 0.37
GRM8 O00222 1/20 0.36
CYP1A2 P05177 1/20 0.36
GRM7 Q14831 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL173553 0.73 PDE2A (0.47) PDE2APDE10AGRM8CYP1A2GRM7
SCHEMBL20698143 0.72 PDE2A (0.36) PDE2APDE10AGRM8CYP1A2GRM7
SCHEMBL1724939 0.71 PDE10A (0.41) PDE2APDE10AGRM8CYP1A2GRM7
SCHEMBL20698179 0.69 PDE10A (0.39) PDE2APDE10AGRM8CYP1A2GRM7
SCHEMBL1725188 0.68 MAPT (0.49)
SCHEMBL24158238 0.68 HSP90AA1 (0.37)
SCHEMBL173584 0.68 PDE10A (0.47) PDE2APDE10AGRM8CYP1A2GRM7
SCHEMBL24158349 0.67 HSP90AA1 (0.37) PDE2A
SCHEMBL20698206 0.67 PDE10A (0.39) PDE2APDE10AGRM8CYP1A2GRM7
SCHEMBL1726288 0.66 PDE2A (0.39) PDE2APDE10AGRM8CYP1A2GRM7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019020981-A1 PYRAZOLE, ISOTHIAZOLE AND ISOXAZOLE DERIVATIVES USEFUL AS AGRICULTURAL FUNGICIDES REDAG CROP PROTECTION LTD. (GB) 2019-01-31 WO disclosed