SCHEMBL20707809

SCHEMBL20707809

O=C(Nc1ccc(C(F)(F)F)cn1)C1CC1

nearest known ligand 0.71

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 1/20 0.71
DEGS1 O15121 3/20 0.62
RAB9A P51151 4/20 0.57
NPC1 O15118 3/20 0.57
PTGS1 P23219 2/20 0.57
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
LMNA P02545 1/20 0.54
POLB P06746 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
ALDH1A1 P00352 2/20 0.53
ABL1 P00519 1/20 0.53
HCRTR1 O43613 2/20 0.51
GAA P10253 1/20 0.50
KDR P35968 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13716370 0.93 NPY5R (0.64) NPY5RDEGS1RAB9ANPC1PTGS1
SCHEMBL13256782 0.85 NPY5R (0.55) NPY5RDEGS1RAB9ANPC1PTGS1
SCHEMBL16422569 0.85 NPY5R (0.55) NPY5RDEGS1RAB9ANPC1PTGS1
SCHEMBL12203141 0.84 NPY5R (0.60) NPY5RDEGS1RAB9ANPC1KMT2A
Velneperit SCHEMBL10114559 0.84 NPY5R (1.00) NPY5RDEGS1RAB9ANPC1PTGS1
SCHEMBL13840438 0.84 NPY5R (0.77) NPY5RDEGS1RAB9ANPC1PTGS1
Velneperit SCHEMBL2806595 0.84 NPY5R (1.00) NPY5RDEGS1RAB9ANPC1PTGS1
Velneperit SCHEMBL29355442 0.84 NPY5R (1.00) NPY5RDEGS1RAB9ANPC1PTGS1
SCHEMBL13840453 0.83 NPY5R (0.75) NPY5RDEGS1RAB9ANPC1PTGS1
SCHEMBL13840450 0.83 NPY5R (0.72) NPY5RDEGS1RAB9ANPC1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2888229-B1 alpha7 NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS AND USES THEREOF MERCK SHARP & DOHME (US) 2019-02-06 EP disclosed