SCHEMBL20733015

SCHEMBL20733015

COC(=O)c1ccc(-c2cncc3ncc(I)cc23)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SGK1 O00141 1/20 0.46
CAMKK2 Q96RR4 1/20 0.46
SLC2A1 P11166 1/20 0.44
EGFR P00533 2/20 0.41
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
NEK1 Q96PY6 3/20 0.39
HPGD P15428 3/20 0.39
MAPK1 P28482 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ATM Q13315 1/20 0.38
CYP11B1 P15538 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20733018 0.85 SGK1 (0.44) SGK1CAMKK2SLC2A1EGFRALDH1A1
SCHEMBL20733083 0.78 HPGD (0.59) ALDH1A1KDM4EHPGDGAA
SCHEMBL20733016 0.74 MELK (0.42) SGK1CAMKK2SLC2A1EGFRHPGD
SCHEMBL31133491 0.72 HTT (0.60) ALDH1A1KDM4EHPGDMAPK1SMN1; SMN2
SCHEMBL18370114 0.72 HTT (0.60) ALDH1A1KDM4EHPGDMAPK1SMN1; SMN2
SCHEMBL10138348 0.71 SLC22A12 (0.51) SGK1CAMKK2SLC2A1EGFRSMN1; SMN2
SCHEMBL20733006 0.71 CCNC (0.51)
SCHEMBL21261147 0.69 EGFR (0.62) SLC2A1EGFRALDH1A1KDM4EMAPT
SCHEMBL2247463 0.68 ATM (0.65) ALDH1A1KDM4EMAPK1GAATDP1
SCHEMBL6909201 0.68 CA1 (0.58) EGFRALDH1A1KDM4EMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666770-A1 NOVEL HETEROCYCLIC COMPOUNDS AS CDK8/19 INHIBITORS Joint Stock Company "Biocad" (RU) 2020-06-17 EP disclosed
WO-2019031990-A1 NOVEL HETEROCYCLIC COMPOUNDS AS CDK8/19 INHIBITORS ЗАКРЫТОЕ АКЦИОНЕРНОЕ ОБЩЕСТВО "БИОКАД" 2019-02-14 WO disclosed