SCHEMBL20734867

SCHEMBL20734867

CC(C)CC1C(=O)CC(=O)N1C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK7 P49862 6/20 0.36
KLK5 Q9Y337 5/20 0.36
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
ABCG2 Q9UNQ0 7/20 0.34
ABCB1 P08183 3/20 0.34
ABCC1 P33527 3/20 0.34
MMP3 P08254 1/20 0.34
ADAM17 P78536 1/20 0.34
MME P08473 1/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
PRSS1 P07477 2/20 0.33
PRSS2 P07478 2/20 0.33
PRSS3 P35030 2/20 0.33
NR1H2 P55055 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20734866 1.00 KLK7 (0.36) KLK7KLK5CHRM2CHRM1CHRM3
SCHEMBL29060299 0.87 KLK7 (0.35) KLK7KLK5CHRM2CHRM1CHRM3
SCHEMBL29526186 0.80 NR1H2 (0.38) KLK7KLK5CHRM2CHRM1CHRM3
SCHEMBL32683207 0.80 CHRM2 (0.35) KLK7KLK5CHRM2CHRM1CHRM3
SCHEMBL34475689 0.79 CHRM2 (0.38) KLK7KLK5CHRM2CHRM1CHRM3
SCHEMBL14515887 0.79 CHRM2 (0.38) KLK7KLK5CHRM2CHRM1CHRM3
SCHEMBL581822 0.79 CHRM2 (0.34) KLK7KLK5CHRM2CHRM1CHRM3
SCHEMBL20734946 0.78 CHRM2 (0.33) KLK7KLK5CHRM2CHRM1CHRM3
SCHEMBL20734945 0.78 CHRM2 (0.33) KLK7KLK5CHRM2CHRM1CHRM3
SCHEMBL3398097 0.78 CHRM2 (0.37) KLK7KLK5CHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019029274-A1 4-OXO-ALKYLATED TETRAMIC ACID COMPOUND AND PREPARATION METHOD THEREFOR 北京卓凯生物技术有限公司 2019-02-14 WO disclosed
WO-2019029273-A1 4-OXO-ALKYLATED TETRAMIC ACID COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 北京卓凯生物技术有限公司 2019-02-14 WO disclosed