SCHEMBL20738562

SCHEMBL20738562

CCn1ncc2c1CN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.43
SLC34A1 Q06495 2/20 0.41
MAPT P10636 2/20 0.41
ESR2 Q92731 1/20 0.40
PIK3CD O00329 5/20 0.40
MAPK1 P28482 1/20 0.40
NAMPT P43490 1/20 0.39
HPGDS O60760 2/20 0.39
HDAC1 Q13547 1/20 0.39
DDB1 Q16531 1/20 0.39
CRBN Q96SW2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9918094 0.87 NR1H2 (0.42) NR1H2SLC34A1MAPTESR2MAPK1
SCHEMBL20392577 0.86 SLC34A1 (0.42) NR1H2SLC34A1MAPTESR2MAPK1
SCHEMBL18493673 0.86 SLC34A1 (0.42) NR1H2SLC34A1MAPTESR2MAPK1
SCHEMBL6891275 0.86 NR1H2 (0.41) NR1H2SLC34A1MAPTESR2MAPK1
SCHEMBL23372979 0.85 NR1H2 (0.40) NR1H2SLC34A1MAPTESR2MAPK1
SCHEMBL17561650 0.85 SLC34A1 (0.49) NR1H2SLC34A1MAPTESR2MAPK1
SCHEMBL19505292 0.85 PIK3CD (0.35) MAPTPIK3CDMAPK1NAMPTHPGDS
SCHEMBL20364274 0.82 NR1H2 (0.46) NR1H2SLC34A1MAPTESR2MAPK1
SCHEMBL5720871 0.82 NR1H2 (0.42) NR1H2SLC34A1MAPTESR2MAPK1
SCHEMBL5720876 0.81 NR1H2 (0.38) NR1H2SLC34A1MAPTESR2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250214977-A1 STAT6 INHIBITORS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2025-07-03 US disclosed
US-11912702-B2 Substituted pyridines as inhibitors of histone deacetylase ALKERMES, INC. (US) 2024-02-27 US disclosed
US-11912702-B2 Substituted pyridines as inhibitors of histone deacetylase ALKERMES, INC. (US) 2024-02-27 US disclosed
EP-3664802-B1 BICYCLIC INHIBITORS OF HISTONE DEACETYLASE ALKERMES INC (US) 2022-02-23 EP disclosed
US-11225475-B2 Substituted pyridines as inhibitors of histone deacetylase ALKERMES, INC. (US) 2022-01-18 US disclosed
US-20210147410-A1 BICYCLIC INHIBITORS OF HISTONE DEACETYLASE JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2021-05-20 US disclosed
WO-2019032528-A1 BICYCLIC INHIBITORS OF HISTONE DEACETYLASE RODIN THERAPEUTICS, INC (US) 2019-02-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210147410-A1 BICYCLIC INHIBITORS OF HISTONE DEACETYLASE HDAC2, HDAC1, HDAC3 NR1H2 150/4885SLC34A1 2659/4885MAPT 1007/4885
US-20250214977-A1 STAT6 INHIBITORS AND USES THEREOF STAT6, STAT5B, STAT5A NR1H2 1135/4885SLC34A1 4204/4885MAPT 3335/4885
US-11225475-B2 Substituted pyridines as inhibitors of histone deacetylase HDAC2, HDAC1, HDAC3 NR1H2 482/4885SLC34A1 1746/4885MAPT 955/4885
US-11912702-B2 Substituted pyridines as inhibitors of histone deacetylase HDAC2, HDAC1, HDAC3 NR1H2 470/4885SLC34A1 1832/4885MAPT 975/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.