SCHEMBL2074092

SCHEMBL2074092

O=C(Nc1cc(N2CCN(C3CCCCC3)CC2)ncn1)N1CCC(F)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.46
RAB9A P51151 2/20 0.46
ALDH1A1 P00352 2/20 0.46
EGFR P00533 2/20 0.42
ERBB3 P21860 2/20 0.42
NPC1 O15118 1/20 0.41
ATM Q13315 1/20 0.41
PDGFRB P09619 1/20 0.41
AXL P30530 1/20 0.40
MERTK Q12866 1/20 0.40
POLB P06746 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
FAAH O00519 1/20 0.39
P4HTM Q9NXG6 1/20 0.39
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2075851 0.99 HRH4 (0.51) HRH4SMN1; SMN2RAB9AALDH1A1EGFR
SCHEMBL2074889 0.92 HRH4 (0.55) HRH4SMN1; SMN2RAB9AALDH1A1EGFR
SCHEMBL2074972 0.92 HRH4 (0.55) HRH4SMN1; SMN2RAB9AALDH1A1EGFR
SCHEMBL2075259 0.92 HRH4 (0.55) HRH4SMN1; SMN2RAB9AALDH1A1EGFR
SCHEMBL2074954 0.92 HRH4 (0.55) HRH4SMN1; SMN2RAB9AALDH1A1EGFR
SCHEMBL2074480 0.92 HRH4 (0.55) HRH4SMN1; SMN2RAB9AALDH1A1EGFR
SCHEMBL2076138 0.91 HRH4 (0.54) HRH4SMN1; SMN2RAB9AALDH1A1EGFR
SCHEMBL2073074 0.90 HRH4 (0.52) HRH4SMN1; SMN2RAB9AALDH1A1EGFR
SCHEMBL2075478 0.90 HRH4 (0.54) HRH4SMN1; SMN2RAB9AALDH1A1PDGFRB
SCHEMBL2075465 0.90 HRH4 (0.52) HRH4SMN1; SMN2RAB9AALDH1A1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7902184-B2 Piperazinyl pyrimidine derivatives HOFFMANN-LA ROCHE INC. (US) 2011-03-08 US claimed
US-7902184-B2 Piperazinyl pyrimidine derivatives HOFFMANN-LA ROCHE INC. (US) 2011-03-08 US disclosed