SCHEMBL20744010

SCHEMBL20744010

CN1C2CCC1CN(Cc1ccc(Nc3ncc(F)cn3)nc1)C2

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 4/20 0.44
CDK2 P24941 1/20 0.44
CDK6 Q00534 17/20 0.42
CDK4 P11802 11/20 0.42
CCND1 P24385 4/20 0.42
CNR2 P34972 1/20 0.41
CCND3 P30281 3/20 0.40
CCNA2 P20248 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23296205 0.88 CDK6 (0.43) CDK1CDK2CDK6CDK4CCND1
SCHEMBL20744720 0.85 CDK6 (0.42) CDK1CDK2CDK6CDK4CCND1
SCHEMBL20744436 0.84 TLR7 (0.40) CDK1CDK2CDK6CDK4CCND1
SCHEMBL29686224 0.81 CCND1 (0.43) CDK1CDK2CDK6CDK4CCND1
SCHEMBL20744431 0.81 CCND1 (0.55) CDK1CDK2CDK6CDK4CCND1
SCHEMBL30579744 0.78 CDK6 (0.58) CDK1CDK2CDK6CDK4CCND1
SCHEMBL20744519 0.78 CDK6 (0.58) CDK1CDK2CDK6CDK4CCND1
SCHEMBL29414480 0.78 CDK6 (0.61) CDK1CDK2CDK6CDK4CCND1
SCHEMBL20744419 0.77 CDK6 (0.49) CDK1CDK2CDK6CDK4CCND1
SCHEMBL20744517 0.76 CDK6 (0.57) CDK1CDK2CDK6CDK4CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019035008-A1 CDK4/6 INHIBITORS AND USE THEREOF BEIJING XUANYI PHARMASCIENCES CO., LTD. (CN) 2019-02-21 WO disclosed