SCHEMBL2074448

SCHEMBL2074448

CC(C)N1CCN(c2ccnc(NC(=O)C3CCCCC3)n2)CC1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.48
HRH4 Q9H3N8 6/20 0.47
OGA O60502 1/20 0.47
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
SHMT2 P34897 1/20 0.43
ALK Q9UM73 3/20 0.42
IGF1R P08069 2/20 0.42
TP53BP1 Q12888 1/20 0.42
CXCR4 P61073 1/20 0.42
GSK3B P49841 1/20 0.41
DYRK1A Q13627 1/20 0.41
ACACB O00763 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2075511 0.99 HRH4 (0.48) IDH1HRH4OGAKDM4EALDH1A1
SCHEMBL2074799 0.84 HRH4 (0.46) IDH1HRH4SHMT2ALKIGF1R
SCHEMBL2075507 0.83 HRH4 (0.47) IDH1HRH4SHMT2ALKIGF1R
SCHEMBL2073765 0.78 HRH4 (0.50) HRH4OGAALDH1A1SHMT2CXCR4
SCHEMBL1089041 0.78 CCR4 (0.52) HRH4KDM4EALDH1A1ALKIGF1R
SCHEMBL2072892 0.77 OGA (0.48) HRH4OGACXCR4
SCHEMBL2072493 0.76 SMN1; SMN2 (0.46) HRH4ALDH1A1GSK3BDYRK1A
SCHEMBL2076140 0.76 OGA (0.47) HRH4OGAALDH1A1GSK3BDYRK1A
SCHEMBL1089742 0.75 HRH4 (0.49) HRH4SHMT2ALKIGF1RCXCR4
SCHEMBL2074665 0.74 KDM4E (0.46) HRH4OGAKDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7902184-B2 Piperazinyl pyrimidine derivatives HOFFMANN-LA ROCHE INC. (US) 2011-03-08 US disclosed