SCHEMBL20754698

SCHEMBL20754698

C=C(/C=C/c1ccc(CC(=O)Nc2ccc(N(C)C)cc2)cc1)c1ncc[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP8 P22894 1/20 0.41
MAPT P10636 5/20 0.41
RECQL P46063 1/20 0.41
GAA P10253 2/20 0.41
GFER P55789 1/20 0.41
MMP13 P45452 3/20 0.40
CACNA1I Q9P0X4 2/20 0.40
KMT2A Q03164 2/20 0.39
LMNA P02545 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
HSD17B3 P37058 1/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
HDAC1 Q13547 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20754456 0.90 CYP1A2 (0.45) MMP8MAPTRECQLGAAGFER
SCHEMBL22733792 0.90 CYP1A2 (0.45) MMP8MAPTRECQLGAAGFER
SCHEMBL20754432 0.89 SMN1; SMN2 (0.49) MAPTGAAKMT2ALMNANPSR1
SCHEMBL20754425 0.89 KMT2A (0.41) MAPTGAAKMT2ALMNANPSR1
SCHEMBL20754460 0.87 SMN1; SMN2 (0.51) MAPTGAAKMT2ALMNAALDH1A1
SCHEMBL20746339 0.79 SMN1; SMN2 (0.51) MAPTRECQLGAAKMT2ALMNA
SCHEMBL20746341 0.79 SMN1; SMN2 (0.51) MAPTRECQLGAAKMT2ALMNA
SCHEMBL20746542 0.78 SMN1; SMN2 (0.52) MAPTGAAKMT2ALMNANPSR1
SCHEMBL20746541 0.78 SMN1; SMN2 (0.52) MAPTGAAKMT2ALMNANPSR1
SCHEMBL20746552 0.77 GAA (0.53) MAPTGAAKMT2ALMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019036607-A1 IMIDAZOLE-BASED ANTICANCER AGENTS AND DERIVATIVES THEREOF, AND METHODS OF MAKING AND USING SAME THE UNIVERSITY OF TOLEDO (US) 2019-02-21 WO disclosed