SCHEMBL2076498

SCHEMBL2076498

CCN1CCN(c2cc(NC(=O)N3CCc4ccccc43)ncn2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.50
USP2 O75604 1/20 0.50
SMN1; SMN2 Q16637 7/20 0.49
NPC1 O15118 6/20 0.49
RAB9A P51151 6/20 0.49
NFKB1 P19838 4/20 0.49
NFKB2 Q00653 4/20 0.49
RELA Q04206 4/20 0.49
TP53 P04637 3/20 0.49
ALDH1A1 P00352 2/20 0.48
PKM P14618 3/20 0.47
HDAC3 O15379 1/20 0.47
ABL1 P00519 1/20 0.47
BCR P11274 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2075728 0.86 SMN1; SMN2 (0.52) MAPTUSP2SMN1; SMN2NPC1RAB9A
SCHEMBL2074775 0.83 HDAC3 (0.50) SMN1; SMN2NPC1ALDH1A1HDAC3ABL1
SCHEMBL2073004 0.77 KIT (0.49) SMN1; SMN2RAB9AALDH1A1HDAC3ABL1
SCHEMBL2075221 0.76 SMN1; SMN2 (0.51) SMN1; SMN2RAB9AALDH1A1HDAC3ABL1
SCHEMBL2075163 0.76 SMN1; SMN2 (0.51) SMN1; SMN2RAB9AALDH1A1HDAC3ABL1
SCHEMBL2075487 0.75 MAPK1 (0.47) MAPTSMN1; SMN2ALDH1A1HDAC3ABL1
SCHEMBL2075182 0.74 KIT (0.46) MAPTSMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL2073422 0.72 KIT (0.45) SMN1; SMN2RAB9AALDH1A1HDAC3ABL1
SCHEMBL2075539 0.72 KIT (0.48) SMN1; SMN2RAB9AALDH1A1HDAC3ABL1
SCHEMBL2072611 0.72 SMN1; SMN2 (0.73) SMN1; SMN2NPC1RAB9AALDH1A1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7902184-B2 Piperazinyl pyrimidine derivatives HOFFMANN-LA ROCHE INC. (US) 2011-03-08 US disclosed