SCHEMBL20780772

SCHEMBL20780772

C=CC(=O)Nc1ccc2ncnc(Nc3ccc(Oc4ccc5cc[nH]c5c4)c(C)c3)c2c1

nearest known ligand 0.67

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.67
FYN P06241 7/20 0.59
SRC P12931 7/20 0.59
ERBB2 P04626 5/20 0.57
ERBB4 Q15303 2/20 0.55
BLK P51451 1/20 0.51
BMX P51813 1/20 0.51
JAK3 P52333 1/20 0.51
BTK Q06187 1/20 0.51
VCP P55072 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22200858 0.89 EGFR (0.61) EGFRFYNSRCERBB2ERBB4
SCHEMBL4463689 0.85 EGFR (0.65) EGFRFYNSRCERBB2ERBB4
SCHEMBL22076859 0.85 EGFR (0.48) EGFRFYNSRCERBB2
SCHEMBL20780771 0.84 EGFR (0.67) EGFRERBB2
SCHEMBL29025870 0.84 EGFR (0.67) EGFRERBB2
SCHEMBL20780983 0.84 EGFR (0.57) EGFRFYNSRCERBB2ERBB4
SCHEMBL7127185 0.81 EGFR (1.00) EGFRFYNSRCERBB2ERBB4
SCHEMBL12888225 0.81 EGFR (0.62) EGFRFYNSRCERBB2ERBB4
SCHEMBL12888646 0.79 EGFR (0.67) EGFRFYNSRCERBB2ERBB4
SCHEMBL12888131 0.79 EGFR (0.59) EGFRFYNSRCERBB2ERBB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3677583-A1 NITROGENOUS HETEROCYCLIC COMPOUND, PREPARATION METHOD, INTERMEDIATE, COMPOSITION, AND APPLICATION Shanghai Pharmaceuticals Holding Co., Ltd. (CN) 2020-07-08 EP disclosed
WO-2019042409-A1 NITROGENOUS HETEROCYCLIC COMPOUND, PREPARATION METHOD, INTERMEDIATE, COMPOSITION, AND APPLICATION 上海医药集团股份有限公司 2019-03-07 WO disclosed