SCHEMBL20780835

SCHEMBL20780835

C=CC(=O)Nc1ccc2ncc(C#N)c(Nc3ccc(Oc4cnc5c(cnn5C)c4)c(C)c3)c2c1

nearest known ligand 0.54

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.54
ERBB2 P04626 14/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20780790 0.88 EGFR (0.49) EGFRERBB2
SCHEMBL20780834 0.86 EGFR (0.70) EGFRERBB2
SCHEMBL20780789 0.85 EGFR (0.55) EGFRERBB2
SCHEMBL4461374 0.85 EGFR (0.67) EGFRERBB2
SCHEMBL4471834 0.79 EGFR (0.58) EGFRERBB2
SCHEMBL20780773 0.78 EGFR (0.80) EGFRERBB2
SCHEMBL30478673 0.78 EGFR (0.80) EGFRERBB2
SCHEMBL4472701 0.78 ERBB2 (0.54) EGFRERBB2
SCHEMBL4464220 0.76 EGFR (0.57) EGFRERBB2
SCHEMBL20395260 0.75 EGFR (0.70) EGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3677583-A1 NITROGENOUS HETEROCYCLIC COMPOUND, PREPARATION METHOD, INTERMEDIATE, COMPOSITION, AND APPLICATION Shanghai Pharmaceuticals Holding Co., Ltd. (CN) 2020-07-08 EP disclosed
WO-2019042409-A1 NITROGENOUS HETEROCYCLIC COMPOUND, PREPARATION METHOD, INTERMEDIATE, COMPOSITION, AND APPLICATION 上海医药集团股份有限公司 2019-03-07 WO disclosed