SCHEMBL20780923

SCHEMBL20780923

C=CC(=O)Nc1ccc2ncnc(Nc3ccc(Oc4cnc5ccnn5c4)c(C)c3)c2c1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.60
ERBB2 P04626 5/20 0.60
FYN P06241 7/20 0.55
SRC P12931 7/20 0.55
BLK P51451 1/20 0.52
BMX P51813 1/20 0.52
JAK3 P52333 1/20 0.52
BTK Q06187 1/20 0.52
ERBB4 Q15303 1/20 0.52
VCP P55072 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22076868 0.86 EGFR (0.59) EGFRERBB2
SCHEMBL29025859 0.84 EGFR (0.84) EGFRERBB2
SCHEMBL20780911 0.84 EGFR (0.84) EGFRERBB2
SCHEMBL4463689 0.84 EGFR (0.65) EGFRERBB2FYNSRCBLK
SCHEMBL12888646 0.83 EGFR (0.67) EGFRERBB2FYNSRCBLK
SCHEMBL22200666 0.82 EGFR (0.60) EGFRERBB2FYNSRCBLK
SCHEMBL20780826 0.82 EGFR (0.59) EGFRERBB2FYNSRCBLK
SCHEMBL12888131 0.81 EGFR (0.59) EGFRERBB2FYNSRCBLK
SCHEMBL20780822 0.81 EGFR (0.59) EGFRERBB2FYNSRCBLK
SCHEMBL12872964 0.80 ERBB2 (0.54) EGFRERBB2ERBB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3677583-A1 NITROGENOUS HETEROCYCLIC COMPOUND, PREPARATION METHOD, INTERMEDIATE, COMPOSITION, AND APPLICATION Shanghai Pharmaceuticals Holding Co., Ltd. (CN) 2020-07-08 EP disclosed
WO-2019042409-A1 NITROGENOUS HETEROCYCLIC COMPOUND, PREPARATION METHOD, INTERMEDIATE, COMPOSITION, AND APPLICATION 上海医药集团股份有限公司 2019-03-07 WO disclosed