SCHEMBL20815331

SCHEMBL20815331

C[C@H](Nc1ncc2c(n1)N(C1CCCC1)CC(C)(C)C(=O)N2C)c1ccccc1F

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 12/20 0.43
IDH1 O75874 7/20 0.40
BRD4 O60885 1/20 0.40
BRDT Q58F21 1/20 0.40
MAPK8 P45983 1/20 0.38
MAPK9 P45984 1/20 0.38
MAPK10 P53779 1/20 0.38
MAPK14 Q16539 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL523461 1.00 PLK1 (0.43) PLK1IDH1BRD4BRDTMAPK8
SCHEMBL523126 1.00 PLK1 (0.43) PLK1IDH1BRD4BRDTMAPK8
SCHEMBL522682 0.89 IDH1 (0.42) PLK1IDH1BRD4BRDT
SCHEMBL522943 0.89 IDH1 (0.42) PLK1IDH1BRD4BRDT
SCHEMBL523913 0.89 PLK1 (0.46) PLK1IDH1BRD4BRDT
SCHEMBL523096 0.89 PLK1 (0.43) PLK1IDH1BRD4BRDT
SCHEMBL524087 0.89 PLK1 (0.46) PLK1IDH1BRD4BRDT
SCHEMBL12694797 0.89 PLK1 (0.43) PLK1IDH1BRD4BRDT
SCHEMBL522605 0.88 IDH1 (0.45) PLK1IDH1BRD4BRDT
SCHEMBL522384 0.88 IDH1 (0.45) PLK1IDH1BRD4BRDT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2356122-B1 PROTEIN KINASE INHIBITORS VERTEX PHARMA (US) 2019-03-20 EP disclosed