SCHEMBL2084301

SCHEMBL2084301

Cc1cnc(CC(CCCN)NC(C)c2ccccn2)c(C)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 13/20 0.55
DUSP3 P51452 1/20 0.33
KMT2A Q03164 1/20 0.33
PTPN11 Q06124 1/20 0.33
SCN8A Q9UQD0 1/20 0.32
GPR142 Q7Z601 2/20 0.32
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
ADORA2B P29275 1/20 0.30
ABCB11 O95342 1/20 0.30
ESR1 P03372 1/20 0.30
CYP1A2 P05177 1/20 0.30
PGR P06401 1/20 0.30
ADRB2 P07550 1/20 0.30
CHRM2 P08172 1/20 0.30
ADRB1 P08588 1/20 0.30
HTR1A P08908 1/20 0.30
ADRA2A P08913 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
NQO2 P16083 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2087023 0.94 CXCR4 (0.52) CXCR4DUSP3KMT2APTPN11SCN8A
SCHEMBL2085127 0.87 CXCR4 (0.52) CXCR4SCN8AHSP90AA1HSP90AB1ABCB11
Hydrochloric Acid SCHEMBL2083504 0.86 CXCR4 (0.51) CXCR4SCN8AHSP90AA1HSP90AB1ABCB11
SCHEMBL2083756 0.83 CXCR4 (0.53) CXCR4GPR142CHRM2
SCHEMBL2084798 0.80 CXCR4 (0.52) CXCR4GPR142HSP90AA1HSP90AB1ABCB11
SCHEMBL2084903 0.80 CXCR4 (0.48) CXCR4SCN8AGPR142ADRB2CHRM2
SCHEMBL2085719 0.80 CXCR4 (0.48) CXCR4KMT2ASCN8ACYP1A2
Hydrochloric Acid SCHEMBL4566243 0.78 HRH1 (0.41) CXCR4CYP1A2
SCHEMBL2083954 0.78 CXCR4 (0.40) CXCR4GPR142HSP90AA1HSP90AB1ABCB11
SCHEMBL2084352 0.78 CXCR4 (0.45) CXCR4GPR142HSP90AA1HSP90AB1ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7863293-B2 CXCR4 chemokine receptor binding compounds GENZYME CORPORATION (US) 2011-01-04 US disclosed