SCHEMBL20848010

SCHEMBL20848010

CCOC(=O)c1cccc(N2N=C(C(F)(F)F)/C(=C/c3ccc(-c4ccc(Cl)c(C(=O)Nc5cccc(OC)c5)c4)o3)C2=O)c1

nearest known ligand 0.72

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
XPA P23025 16/20 0.72
ERO1A Q96HE7 2/20 0.52
KDM1A O60341 1/20 0.52
MAOA P21397 1/20 0.52
MAOB P27338 1/20 0.52
MEN1 O00255 1/20 0.52
APEX1 P27695 1/20 0.52
NTSR1 P30989 1/20 0.52
GALK1 P51570 1/20 0.52
KMT2A Q03164 1/20 0.52
EP300 Q09472 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20840330 1.00 XPA (0.72) XPAERO1AKDM1AMAOAMAOB
SCHEMBL20840331 1.00 XPA (0.72) XPAERO1AKDM1AMAOAMAOB
SCHEMBL20840292 0.92 XPA (0.83) XPAERO1AKDM1AMAOAMAOB
SCHEMBL29385593 0.92 XPA (0.85) XPAMEN1APEX1NTSR1GALK1
SCHEMBL20840291 0.92 XPA (0.83) XPAERO1AKDM1AMAOAMAOB
SCHEMBL20848012 0.92 XPA (0.83) XPAERO1AKDM1AMAOAMAOB
SCHEMBL19654076 0.92 XPA (0.85) XPAMEN1APEX1NTSR1GALK1
SCHEMBL20840344 0.88 XPA (0.73) XPAERO1AKDM1AMAOAMAOB
SCHEMBL20840345 0.88 XPA (0.73) XPAERO1AKDM1AMAOAMAOB
SCHEMBL22219633 0.88 XPA (0.73) XPAERO1AKDM1AMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3684354-B1 XPA INHIBITOR COMPOUNDS AND THEIR USE UNIV INDIANA RES & TECH CORP (US) 2023-11-15 EP disclosed
US-11207296-B2 XPA inhibitor compounds and their use INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2021-12-28 US disclosed
US-20200222367-A1 XPA INHIBITOR COMPOUNDS AND THEIR USE INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION 2020-07-16 US disclosed
WO-2019060260-A1 XPA INHIBITOR COMPOUNDS AND THEIR USE INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2019-03-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200222367-A1 XPA INHIBITOR COMPOUNDS AND THEIR USE XPOT, XPA, ERCC4 XPA 2/4885ERO1A 926/4885KDM1A 2277/4885
US-11207296-B2 XPA inhibitor compounds and their use XPOT, XPA, ERCC4 XPA 2/4885ERO1A 926/4885KDM1A 2277/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.