SCHEMBL20848655

SCHEMBL20848655

COC(=O)c1ccnc2cc(Cc3cc(Cl)c(Cl)c(Cl)c3C)[nH]c12

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 10/20 0.53
KDM5A P29375 14/20 0.51
KDM5B Q9UGL1 13/20 0.51
KDM4A O75164 7/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16157370 0.85 KDM5A (0.65) KDM4CKDM5AKDM5BKDM4A
SCHEMBL16149757 0.84 KDM4C (0.58) KDM4CKDM5AKDM5BKDM4A
SCHEMBL16150890 0.83 KDM4C (0.76) KDM4CKDM5AKDM5BKDM4A
SCHEMBL16157405 0.80 KDM5A (0.77) KDM4CKDM5AKDM5BKDM4A
SCHEMBL16157410 0.80 KDM5A (0.78) KDM4CKDM5AKDM5BKDM4A
SCHEMBL16157404 0.80 KDM5A (0.76) KDM4CKDM5AKDM5BKDM4A
SCHEMBL17889779 0.79 KDM5A (0.64) KDM4CKDM5AKDM5BKDM4A
SCHEMBL16157333 0.77 KDM5A (0.64) KDM4CKDM5AKDM5BKDM4A
SCHEMBL16149776 0.77 KDM5A (0.83) KDM4CKDM5AKDM5BKDM4A
SCHEMBL16157397 0.77 KDM5A (0.62) KDM4CKDM5AKDM5BKDM4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190092771-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2019-03-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190092771-A1 HISTONE DEMETHYLASE INHIBITORS KDM1B, KDM1A, KDM5A KDM4C 12/4885KDM5A 3/4885KDM5B 6/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.