SCHEMBL20852080

SCHEMBL20852080

CC(C)(C)c1ccc(C(=O)Nc2cccc(CCC(=O)O)c2)c(NC(=O)c2ccc(-c3cccs3)cc2)c1

nearest known ligand 0.71

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 15/20 0.71
PPARD Q03181 7/20 0.71
PPARG P37231 7/20 0.68
PPARA Q07869 5/20 0.68
HSPH1 Q92598 1/20 0.55
ITGB3 P05106 1/20 0.49
ITGA2B P08514 1/20 0.49
HDAC1 Q13547 2/20 0.47
GPBAR1 Q8TDU6 1/20 0.47
MMP2 P08253 1/20 0.46
MMP10 P09238 1/20 0.46
MMP9 P14780 1/20 0.46
MMP8 P22894 1/20 0.46
MMP12 P39900 1/20 0.46
MMP13 P45452 1/20 0.46
MMP14 P50281 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20839733 0.87 NR1H4 (0.72) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839687 0.83 NR1H4 (1.00) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839629 0.78 NR1H4 (0.56) NR1H4PPARDPPARGPPARAHDAC1
SCHEMBL20852079 0.76 NR1H4 (0.81) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839658 0.74 NR1H4 (0.71) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL3875270 0.73 TRPV1 (0.61) HDAC1
SCHEMBL4579561 0.73 HDAC1 (0.71) HDAC1
SCHEMBL20839731 0.73 NR1H4 (0.80) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL4578962 0.73 HDAC1 (0.79) HDAC1
SCHEMBL4580580 0.71 HDAC1 (0.55) HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019057969-A1 DUAL AGONISTS OF FXR AND PPARδ AND THEIR USES Johann Wolfgang Goethe-Universität (DE) 2019-03-28 WO disclosed