SCHEMBL20858951

SCHEMBL20858951

COc1cc(C)c(CN2CCCCC2)c(O)c1C(=O)/C=C/c1cccc(C)c1

nearest known ligand 0.71

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 12/20 0.51
MAPT P10636 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7030123 0.93 ABCB1 (0.57) ABCB1
SCHEMBL20858957 0.92 ABCB1 (0.59) ABCB1
SCHEMBL20858997 0.91 ABCB1 (0.57) ABCB1MAPT
SCHEMBL20858993 0.91 ABCB1 (0.60) ABCB1
SCHEMBL7026331 0.90 ABCB1 (0.49) ABCB1MAPTNPSR1
SCHEMBL20858964 0.89 ABCB1 (0.49) ABCB1MAPTNPSR1
SCHEMBL20858974 0.87 ABCB1 (0.57) ABCB1MAPT
SCHEMBL20858975 0.86 ABCB1 (0.47) ABCB1MAPTNPSR1
SCHEMBL744982 0.84 ABCB1 (0.62) ABCB1MAPT
SCHEMBL746215 0.84 ABCB1 (0.67) ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2429292-B1 COMPOUNDS AND COMPOSITIONS COMPRISING CDK INHIBITORS AND THEIR USE IN THE TREATMENT OF CANCER GEORGIA STATE UNIV RESEARCH FOUNDATION (US) 2019-04-03 EP disclosed