SCHEMBL20895751

SCHEMBL20895751

COc1cc(-c2ccn3c(-c4cccc(N(OC=O)C(=O)NCC(F)(F)F)c4)cnc3c2)ncn1

nearest known ligand 0.68

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KDR P35968 19/20 0.68
FGFR3 P22607 19/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11908501 0.89 FGFR3 (0.68) KDRFGFR3
SCHEMBL11909507 0.87 KDR (0.65) KDRFGFR3
SCHEMBL11909474 0.87 FGFR3 (0.66) KDRFGFR3
SCHEMBL3322879 0.86 FGFR3 (0.54) KDRFGFR3
SCHEMBL3324434 0.86 FGFR3 (0.52) KDRFGFR3
SCHEMBL20895722 0.85 KDR (0.66) KDRFGFR3
SCHEMBL11907993 0.84 FGFR3 (0.65) KDRFGFR3
SCHEMBL11908369 0.84 KDR (0.67) KDRFGFR3
SCHEMBL11908090 0.84 FGFR3 (0.68) KDRFGFR3
SCHEMBL11909121 0.84 FGFR3 (0.68) KDRFGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2300465-B1 IMIDAZOPYRIDINE DERIVATIVES AS INHIBITORS OF RECEPTOR TYROSINE KINASES ASTEX THERAPEUTICS LTD (GB) 2019-04-17 EP disclosed