SCHEMBL20909042

SCHEMBL20909042

C[C@H]1CC2(CCN(c3ncc(-c4c(O)ccc(Cl)c4Cl)nc3CO)CC2)CO1

nearest known ligand 0.71

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 20/20 0.71
KCNH2 Q12809 2/20 0.39
EGFR P00533 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20909050 0.94 PTPN11 (0.69) PTPN11KCNH2EGFR
SCHEMBL20909377 0.90 PTPN11 (0.60) PTPN11KCNH2EGFR
SCHEMBL22594986 0.90 PTPN11 (0.66) PTPN11KCNH2EGFR
SCHEMBL20909056 0.85 PTPN11 (0.68) PTPN11KCNH2EGFR
SCHEMBL30787825 0.83 PTPN11 (1.00) PTPN11KCNH2EGFR
SCHEMBL20899360 0.83 PTPN11 (1.00) PTPN11KCNH2EGFR
SCHEMBL20909035 0.82 PTPN11 (0.73) PTPN11KCNH2
SCHEMBL20909053 0.81 PTPN11 (0.50) PTPN11KCNH2EGFR
SCHEMBL20909371 0.79 PTPN11 (0.72) PTPN11KCNH2
SCHEMBL20909043 0.78 PTPN11 (0.72) PTPN11KCNH2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019075265-A1 PYRIDINE, PYRAZINE, AND TRIAZINE COMPOUNDS AS ALLOSTERIC SHP2 INHIBITORS Revolution Medicines, Inc. (US) 2019-04-18 WO disclosed